Umbhali: Janice Evans
Umhla Wokudalwa: 1 Eyekhala 2021
Hlaziya Umhla: 23 Isilimela 2024
Anonim
Ranolazine - Side Effects, Mechanism of Action, and Indications
Ividiyo: Ranolazine - Side Effects, Mechanism of Action, and Indications

Umxholo

I-Ranolazine isetyenziswa yodwa okanye namanye amayeza ukunyanga i-angina engapheliyo (iintlungu zesifuba eziqhubekayo okanye uxinzelelo oluvakalayo xa intliziyo ingafumani oksijini yaneleyo). I-Ranolazine ikwiklasi yamayeza abizwa ngokuba yi-anti-anginals. Eyona ndlela isebenza ngayo i-ranolazine ayaziwa ngeli xesha.

I-Ranolazine iza njengokukhutshwa okwandisiweyo (ukusebenza ixesha elide) ithebhulethi ukuthatha ngomlomo. Ihlala ithathwa kunye okanye ngaphandle kokutya kabini imihla ngemihla. Thatha i-ranolazine ngamaxesha afanayo yonke imihla. Landela izikhokelo kwileyibhile yakho yonyango ngononophelo, kwaye ubuze ugqirha wakho okanye usokhemesti ukuba achaze nayiphi na indawo ongayiqondiyo. Thatha i-ranolazine kanye njengoko kuyalelwe. Musa ukuthatha ngaphezulu okanye ngaphantsi kwayo okanye uthathe rhoqo kunokuba umiselwe ngugqirha wakho.

Ginya iipilisi ngokupheleleyo; musa ukuwaphula, ungawuhlafuna, okanye uwaqhekeze.

Ugqirha wakho uya kuqala ngedosi ephantsi ye-ranolazine kwaye ngokuthe ngcembe andise idosi yakho.

Musa ukuthatha i-ranolazine ukunyanga uhlaselo lwe-angina ngequbuliso. Ugqirha wakho uza kukuxelela into ekufuneka uyenzile ukuba ufumana uhlaselo lwe-angina. Qiniseka ukuba uyayiqonda le ndlela.


I-Ranolazine inokunceda ukulawula imeko yakho kodwa ayizukuyinyanga. Qhubeka nokuthatha i-ranolazine nokuba uziva uphilile. Sukuyeka ukuthatha i-ranolazine ungakhange uthethe nogqirha wakho.

Buza usokhemesti okanye ugqirha wakho ngekopi yolwazi lomenzi wesigulana.

Eli yeza linokumiselwa ezinye izinto; buza ugqirha wakho okanye usokhemesti ngolwazi oluthe kratya.

Ngaphambi kokuba uthathe i-ranolazine,

  • xelela ugqirha wakho kunye nosokhemesti ukuba ngaba uxabana ne-ranolazine, nawaphi na amanye amayeza, okanye naziphi na izithako kwiipilisi zokukhupha i-ranolazine. Buza usokhemesti wakho uluhlu lwezithako.
  • xelela ugqirha wakho ukuba ngaba uthatha nawaphi na amayeza alandelayo: ii-antifungals ezifana ne-itraconazole (Onmel, Sporanox) kunye ne-ketoconazole (Nizoral); i-clarithromycin (i-Biaxin, kwi-Prevpac); amayeza okunyanga intsholongwane kaGawulayo (i-HIV) okanye i-immunodeficiency syndrome (i-AIDS) efana ne-indinavir (Crixivan), lopinavir kunye ne-ritonavir (Kaletra); i-nelfinavir (iViracept), i-ritonavir (i-Norvir, e-Kaletra, e-Viekira Pak, abanye), kunye ne-saquinavir (i-Invirase); nefazodone; amayeza okubanjwa njenge carbamazepine (Carbatrol, Equetro, Tegretol, abanye), phenobarbital, kunye ne phenytoin (Dilantin, Phenytek); irifabutin (Mycobutin); irifampin (Rifadin, Rimactane, eRifamate, eRifater); Kunye nerifapentin (Priftin). Xelela ugqirha wakho ukuba uthatha i-wort yaseSt. Ugqirha wakho unokukuxelela ukuba ungathathi i-ranolazine ukuba uthatha elinye okanye nangaphezulu kula mayeza okanye iimveliso zamayeza.
  • xelela ugqirha wakho kunye nosokhemesti ukuba loluphi olunye amayeza amiselweyo kunye nalawo angabhalwanga, iivithamini, izongezo zesondlo, kunye nemveliso yamayeza owathathayo okanye oceba ukuyithatha. Qiniseka ukuba ukhankanya nayiphi na kwezi zilandelayo: amiodarone (Cordarone, Nexterone, Pacerone); antidepressants ezifana amitriptyline, clomipramine (Anafranil), kunye desipramine (Norpramin); kunye ne-imipramine (Tofranil); amayeza okunyanga i-cholesterol ephezulu njenge-atorvastatin (Lipitor, eCaduet), lovastatin (Altoprev, kwi-Advicor), kunye ne-simvastatin (iZocor, eSimcor, eVytorin); icyclosporine (Gengraf, Neoral, Sandimmune); idigoxin (Lanoxin); diltiazem (Cardizem, Dilacor, Tiazac, nabanye); dofetilide; (ITikosyn); i-erythromycin (i-EES, i-Erythrocin, i-PCE); i-fluconazole (iDiflucan); amayeza esigulo sengqondo njenge-haloperidol (Haldol), risperidone (Risperdal), thioridazine, kunye ne-ziprasidone (Geodon); metformin (Fortamet, Glumetza, kwiGlucovance, abanye); quinidine (kwiNuedexta); i-sirolimus (iRapamune); i-sotalol (iBetapace, iSorine); itacrolimus (Astagraf, Envarsus XR, Prograf); kunye ne-verapamil (Calan, Covera, Verelan, abanye). Ugqirha wakho unokufuna ukutshintsha amayeza akho okanye akubeke esweni ngononophelo kwiziphumo ebezingalindelekanga. Amanye amayeza amaninzi anokusebenzisana ne-ranolazine, ke qiniseka ukuxelela ugqirha wakho malunga nawo onke amayeza owathathayo, nkqu nalawo angaveli kolu luhlu okanye kuluhlu olungentla.
  • xelela ugqirha wakho ukuba ukhe unesifo sesibindi. Ugqirha wakho angakuxelela ukuba awufanele uthathe i-ranolazine.
  • xelela ugqirha wakho ukuba wena okanye nabani na kusapho lwakho unethuba elide le-QT (ingxaki yentliziyo enqabileyo enokubangela ukuba utyhafe okanye ukubetha kwentliziyo ngokungaqhelekanga) okanye ukubetha kwentliziyo okukhawulezayo, okucothayo, okanye okungaqhelekanga. Xelela ugqirha wakho ukuba unayo okanye wakha wanayo i-electrocardiogram engaqhelekanga (i-ECG: uvavanyo olurekhoda umsebenzi wombane wentliziyo), amanqanaba asezantsi e-potassium egazini, okanye isifo sezintso.
  • xelela ugqirha wakho ukuba ukhulelwe, cwangcisa ukukhulelwa, okanye uncancisa. Ukuba ukhulelwa ngelixa uthatha i-ranolazine, tsalela ugqirha wakho.
  • Kuya kufuneka uyazi ukuba i-ranolazine inokukwenza ube nesiyezi kwaye ube nentloko elula. Musa ukuqhuba imoto, ukusebenzisa oomatshini, okanye ukuthatha inxaxheba kwimisebenzi efuna ukuphapha kwengqondo kunye nokulungelelanisa de ube uyazi ukuba lonyango lukuchaphazela njani.

Musa ukusela ijusi yeziqhamo ze grapefruit okanye utye iimveliso ze grapefruit ngelixa uthatha eli yeza.


Tsiba idosi ephosiweyo kwaye uqhubeke neshedyuli yakho yesiqhelo yokulinganisa Sukuthatha idosi ephindwe kabini ukwenza eyilahlekileyo.

I-Ranolazine inokubangela iziphumo ebezingalindelekanga. Tshela ugqirha wakho ukuba ngaba ezinye zeempawu zinzima okanye azihambi:

  • isicaphucaphu
  • ukuqhina
  • intloko ebuhlungu
  • isiyezi

Ezinye iziphumo ebezingalindelekanga zinokuba nzulu. Ukuba ufumana nayiphi na le mpawu, biza ugqirha wakho ngokukhawuleza:

  • ngokukhawuleza, ukubetha, okanye ukubetha kwentliziyo okungaqhelekanga
  • ubunzima bokuphefumla
  • isiqaqa

I-Ranolazine inokubangela ezinye iziphumo ebezingalindelekanga. Biza ugqirha wakho ukuba unengxaki engaqhelekanga ngelixa uthatha eli yeza.

Gcina eli yeza kwisikhongozeli lifikile, livalekile, kwaye alifumaneki ebantwaneni. Yigcine kubushushu begumbi kwaye kude nobushushu obuninzi kunye nokufuma (hayi kwigumbi lokuhlambela).

Amayeza angafunekiyo kufuneka achithwe ngeendlela ezizodwa zokuqinisekisa ukuba izilwanyana zasekhaya, abantwana kunye nabanye abantu abanakuzisebenzisa. Nangona kunjalo, akufuneki uligungxule eli yeza kwindlu yangasese. Endaweni yoko, eyona ndlela yokulahla amayeza akho yinkqubo yokubuyisa amayeza. Thetha kumayeza wakho okanye unxibelelane nesebe lakho lenkunkuma / lokurisayikilisha ukuze ufunde malunga neenkqubo zokubuyisa kwindawo ohlala kuyo. Jonga i-FDA's Safe Disposal of Medicines website (http://goo.gl/c4Rm4p) ngolwazi oluthe kratya ukuba awunakho ukufikelela kwinkqubo yokubuyisa.


Kubalulekile ukugcina onke amayeza ngaphandle kwamehlo kunye nokufikelela kwabantwana njengezikhongozeli ezininzi (ezinje ngeeveki zeepilisi zeveki kunye nezo zamehlo, iikhrim, iipatches, kunye ne-inhalers) azinyangeki kwaye abantwana abancinci banokuzivula ngokulula. Ukukhusela abantwana abancinci kwiityhefu, soloko ukhiya iminqwazi yokhuseleko kwaye ubeke amayeza kwindawo ekhuselekileyo-leyo iphakame kwaye iphakame kwaye ingabonakali kubo kwaye ifikelele kuyo. http://www.upandaway.org

Kwimeko yokugqithisa, fowunela umnxeba wolawulo lwetyhefu kwi-1-800-222-1222. Ulwazi lukwafumaneka kwi-Intanethi kwi-https: //www.poisonhelp.org/help. Ukuba ixhoba liye lawa, laxhuzula, linengxaki yokuphefumla, okanye alikwazi ukuvuswa, ngoko nangoko lifowunele iinkonzo zongxamiseko ngo-911.

Iimpawu libanda kungaquka oku kulandelayo:

  • isicaphucaphu
  • ukugabha
  • isiyezi
  • ukudideka
  • umbono kabini
  • iintlungu, ukutshisa, ukuba ndindisholo, okanye ukubetha kulo naliphi na ilungu lomzimba
  • isiqaqa
  • ukushukuma okungalawulekiyo kwilungu lomzimba
  • kunzima ukuthetha
  • ukubona izinto okanye ukuva amazwi angekhoyo

Gcina lonke ixesha lokudibana nogqirha wakho.

Musa ukuvumela nabani na ukuba athathe amayeza akho. Buza usokhemesti wakho nayiphi na imibuzo onayo malunga nokuzalisa amayeza akho.

Kubalulekile ukuba ugcine uluhlu olubhaliweyo lwawo onke amayeza owasebenzisayo amayeza owasebenzisayo, kunye nezinye iimveliso ezinjengeevithamini, iiminerali, okanye ezinye izongezo zokutya. Kuya kufuneka uze nolu luhlu qho xa undwendwela ugqirha okanye ungeniswe esibhedlele. Kukwabalulekile ulwazi ukuba uphathe nawe xa kukho imeko kaxakeka.

  • URanexa®
Ukuhlaziywa kokugqibela-01/15/2016

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