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Inaliti yeRolapitant ayisasebenzi eMelika.

Inaliti ye-Rolapitant isetyenziswa kunye namanye amayeza ukuthintela isicaphucaphu kunye nokugabha okunokwenzeka kwiintsuku ezininzi emva kokufumana amayeza athile e-chemotherapy. I-Rolapitant ikudidi lwamayeza abizwa ngokuba yi-antiemetics. Isebenza ngokuthintela isenzo se-neurokinin kunye ne-P, izinto zendalo kwingqondo ezibangela isicaphucaphu kunye nokugabha.

Inaliti ye-Rolapitant iza njengesisombululo (ulwelo) ukuze ifakwe ngaphakathi ngaphakathi (emthanjeni) ngumboneleli wezempilo esibhedlele okanye ekliniki. Ihlala ifakwa ngaphakathi ngaphakathi njengethamo elinye ngaphezulu kwemizuzu engama-30 kwisithuba seeyure ezimbini ngaphambi kokuqala kwekhemotherapy.

Inaliti ye-Rolapitant inokubangela iimpendulo ezinzulu ngexesha lokufakwa kweyeza, rhoqo kwimizuzu yokuqala. Ugqirha okanye umongikazi uya kukujonga ngononophelo ngelixa ufumana amayeza. Ukuba ufumana naziphi na kwezi mpawu zilandelayo, xelela ugqirha ngokukhawuleza: irhashalala; ukugungxula; ukurhawuzelela; ubunzima bokuphefumla okanye ukugwinya; ukuqhawukelwa ngumphefumlo; ukudumba kwamehlo, ubuso, umlomo, ulwimi, okanye umqala; iintlungu zesifuba; isisu esibuhlungu okanye ukubamba; ukugabha; isiyezi; okanye isiqaqa.


Buza usokhemesti okanye ugqirha wakho ngekopi yolwazi lomenzi wesigulana.

Eli yeza linokumiselwa ezinye izinto; buza ugqirha wakho okanye usokhemesti ngolwazi oluthe kratya.

Ngaphambi kokufumana inaliti yokuqengqeleka,

  • xelela ugqirha wakho kunye nosokhemesti ukuba ngaba uxabisa kwi-rolapitant; nawaphi na amanye amayeza; oyile yeembotyi zesoya; iimbotyi ezinjengeembotyi, amandongomane, ii-ertyisi, okanye iilentile; okanye nasiphi na isithako esenziwe ngenaliti yokuqengqeleka. Buza usokhemesti wakho uluhlu lwezithako.
  • xelela ugqirha wakho ukuba uthatha i-thioridazine okanye ipimozide (Orap). Ugqirha wakho ngekhe afune ukuba ufumane inaliti yokuthambisa ukuba uthatha elinye okanye ngaphezulu kwala mayeza.
  • xelela ugqirha wakho kunye nosokhemesti ukuba loluphi olunye amayeza amiselweyo kunye nalawo angabhalwanga, iivithamini, izongezo zesondlo, kunye nemveliso yamayeza owathathayo okanye oceba ukuyithatha. Qiniseka ukuba ukhankanya nayiphi na kwezi zinto zilandelayo: dextromethorphan (Robitussin, abanye), digoxin (Lanoxin), irinotecan (Camptosar), methotrexate (Otrexup, Rasuvo, Trexall), rifampin (Rifadin, Rimactane, eRifamate, eRifater), rosuvastatin ICrestor), kunye ne-topotecan (Hycamtin). Ugqirha wakho unokufuna ukutshintsha amayeza akho okanye akubeke esweni ngononophelo kwiziphumo ebezingalindelekanga. Amanye amayeza amaninzi anokusebenzisana ne-rolapitant, ke qiniseka ukuxelela ugqirha wakho malunga nawo onke amayeza owathathayo, nkqu nalawo angaveli kolu luhlu.
  • xelela ugqirha wakho ukuba ukhe unesifo sesibindi.
  • xelela ugqirha wakho ukuba ukhulelwe, cwangcisa ukukhulelwa, okanye uncancisa. Ukuba ukhulelwe ngelixa ufumana inaliti yokuqunjelwa, biza ugqirha.

Inaliti ye-Rolapitant inokubangela iziphumo ebezingalindelekanga. Tshela ugqirha wakho ukuba ngaba ezinye zeempawu zinzima okanye azihambi:

  • hiccups
  • isisu esibuhlungu
  • ukunciphisa ukutya
  • isiyezi
  • isilungulela
  • izilonda zomlomo

Ezinye iziphumo ebezingalindelekanga zinokuba nzulu. Ukuba unazo naziphi na kwezi mpawu, biza ugqirha ngokukhawuleza okanye ufumane unyango olungxamisekileyo:

  • umkhuhlane, ukugodola, umqala obuhlungu, okanye ezinye iimpawu zosulelo

Inaliti ye-Rolapitant inokubangela ezinye iziphumo ebezingalindelekanga. Biza ugqirha wakho ukuba unengxaki engaqhelekanga ngelixa uthatha eli yeza.


Ukuba uhlangabezana neziphumo ebezingalindelekanga ezimandundu, wena okanye ugqirha wakho ungathumela ingxelo kwiNkqubo yoKutya kunye nezoLawulo (i-FDA) yeMedWatch yeNkqubo yokuNgxelo ngezeMeko eziGwenxa kwi-Intanethi (http://www.fda.gov/Safety/MedWatch) okanye ngomnxeba ( 1-800-332-1088).

Kwimeko yokugqithisa, fowunela umnxeba wolawulo lwetyhefu kwi-1-800-222-1222. Ulwazi lukwafumaneka kwi-Intanethi kwi-https: //www.poisonhelp.org/help. Ukuba ixhoba liye lawa, laxhuzula, linengxaki yokuphefumla, okanye alikwazi ukuvuswa, ngoko nangoko lifowunele iinkonzo zongxamiseko ngo-911.

Gcina lonke ixesha lokudibana nogqirha wakho.

Kubalulekile ukuba ugcine uluhlu olubhaliweyo lwawo onke amayeza owasebenzisayo amayeza owasebenzisayo, kunye nezinye iimveliso ezinjengeevithamini, iiminerali, okanye ezinye izongezo zokutya. Kuya kufuneka uze nolu luhlu qho xa undwendwela ugqirha okanye ungeniswe esibhedlele. Kukwabalulekile ulwazi ukuba uphathe nawe xa kukho imeko kaxakeka.

  • Varubi®
Ukuhlaziywa kokugqibela-09/15/2020


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