Umbhali: Morris Wright
Umhla Wokudalwa: 23 Utshazimpuzi 2021
Hlaziya Umhla: 1 Utshazimpuzi 2025
Anonim
Flumazenil
Ividiyo: Flumazenil

Umxholo

IFlumazenil liyeza elitofwayo elisetyenziswa esibhedlele ukubuyisela umva ifuthe le-benzodiazepines, eliqela leziyobisi ezinokuthomalalisa, ukulala, ukuxhalabisa, ukuxola kwezihlunu kunye ne-anticonvulsant effect.

Ke, i-flumazenil isetyenziswa ngokubanzi emva kwe-anesthesia yokuvusa abaguli okanye kwimeko yokunxila ngokusetyenziswa gwenxa kwamayeza, umzekelo.

Eli yeza inokufumaneka ngohlobo lwegeneric, kodwa ikwaveliswa ziilabhoratri zaseRoche phantsi kwegama lorhwebo iLanexat. Nangona kunjalo, inokusetyenziswa kuphela ezibhedlele, ingathengiswa kwiikhemesti eziqhelekileyo.

Amanye amagama orhwebo

Ukongeza kwiLanexat, i-flumazenil ikwaveliswa ngamanye amagumbi elebhu kwaye inokuthengiswa phantsi kwamanye amagama orhwebo, anje ngeFlumazenil, Flunexil, Lenazen okanye Flumazil, umzekelo.


Ingaba isebenza kanjani

I-Flumazenil yinto ebophelela kwii-benzodiazepine receptors, ukuthintela ezinye iziyobisi, ezinje ngokudambisa kunye ne-anxiolytics, ekubeni zikwazi ukubopha. Ngale ndlela, amanye amachiza ayayeka ukusebenza, kuba kufuneka azibophelele kwezi receptors ukuze zisebenze.

Ke, i-flumazenil iyakwazi ukuthintela ukusebenza kwamachiza e-benzodiazepine ngaphandle kokuchaphazela ifuthe lamanye amayeza angekho kweli qela.

Yenzelwe ntoni

I-Flumazenil iboniswa ukuba iphazamisa ifuthe lamayeza e-benzodiazepine emzimbeni, yiyo loo nto isetyenziswa kakhulu ukumisa ifuthe le-anesthesia ngokubanzi okanye ukunyanga ukunxila okubangelwa ngamayeza aphezulu e-benzodiazepines.

Kusetyenziswa kwanjani

I-Flumazenil kufuneka isetyenziswe kuphela ziingcali zezempilo esibhedlele, kwaye idosi kufuneka ihlale iboniswa ngugqirha, ngokwale ngxaki kufuneka inyangwe kunye neempawu ezizisiweyo.

Iziphumo ebezingalindelekanga ezinokwenzeka

Ezinye zeziphumo ebezingalindelekanga eziqhelekileyo ze-flumazenil zibandakanya isicaphucaphu, ukugabha, ukubetha kwentliziyo, ixhala kunye noloyiko.


Ngubani ongafanele asebenzise

Esi sixhobo siyaphikiswa kubantu abanezigulo ze-aleji kuwo nawaphi na amacandelo efomula okanye kwizigulana ezifumana unyango lwezifo ezinokubulala i-benzodiazepines.

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