Umbhali: Clyde Lopez
Umhla Wokudalwa: 22 Eyekhala 2021
Hlaziya Umhla: 1 Eyekhala 2024
Anonim
Ziprasidone Pharmacology
Ividiyo: Ziprasidone Pharmacology

Umxholo

Izifundo zibonise ukuba abantu abadala abanesifo sengqondo esixhalabisayo (ukuphazamiseka kwengqondo okuchaphazela ukukhumbula, ukucinga ngokucacileyo, ukunxibelelana, nokwenza imisebenzi yemihla ngemihla kwaye kunokubangela utshintsho kwiimvakalelo nakubuntu) abathatha ii-antipsychotic (amayeza esigulo sengqondo) njenge-ziprasidone banengozi enkulu yokufa ngexesha lonyango. Abantu abadala abanesifo sengqondo esixhalabisayo banokuba nethuba elikhulu lokuba nesifo sokubethwa okanye ukubetha kancinci ngexesha lonyango.

I-Ziprasidone ayivunywanga yi-Food and Drug Administration (FDA) kunyango lweengxaki zokuziphatha kubantu abadala abanesifo sengqondo esixhalabisayo. Thetha nogqirha okumisele la mayeza ukuba wena, ilungu losapho, okanye umntu omkhathalelayo unesifo sengqondo esixhalabisayo kwaye uthatha i-ziprasidone. Ngolwazi oluthe kratya ndwendwela iwebhusayithi ye-FDA: http://www.fda.gov/Drugs

I-Ziprasidone isetyenziselwa ukunyanga iimpawu ze-schizophrenia (isifo sengqondo esibangela ukuphazamiseka okanye ukucinga okungaqhelekanga, ukuphelelwa ngumdla ebomini, kunye neemvakalelo ezinamandla okanye ezingalunganga). Isetyenziselwa ukunyanga iziqendu ze-mania (frenzied, imdaka engaqhelekanga okanye imeko ecaphukisayo) okanye iziqendu ezixubeneyo (iimpawu ze-mania kunye noxinzelelo ezenzeka kunye) kwizigulana ezinesifo se-bipolar (isifo sokudakumba komntu; isifo esibangela iziqendu zoxinzelelo, iziqendu yemania, kunye nezinye iimeko ezingaqhelekanga). I-Ziprasidone ikudidi lwamayeza abizwa ngokuba yi-atypical antipsychotic. Isebenza ngokutshintsha umsebenzi wezinto ezithile zendalo kwingqondo.


I-Ziprasidone iza njengepilisi yokuthatha ngomlomo. Ihlala ithathwa kabini ngemini ngokutya. Thatha i-ziprasidone ngeenxa zonke ngamaxesha afanayo yonke imihla. Landela izikhokelo kwileyibhile yakho yonyango ngononophelo, kwaye ubuze ugqirha wakho okanye usokhemesti ukuba achaze nayiphi na indawo ongayiqondiyo. Thatha i-ziprasidone ngokuchanekileyo njengoko kuyalelwe. Musa ukuthatha ngaphezulu okanye ngaphantsi kwayo okanye uthathe rhoqo kunokuba umiselwe ngugqirha wakho.

Ugqirha wakho unokukuqala kwidosi ephantsi ye-ziprasidone kwaye ngokuthe ngcembe wandise idosi yakho.

I-Ziprasidone inokunceda ukulawula iimpawu zakho kodwa ayizukuyinyanga imeko yakho. Ingathatha iiveki ezimbalwa okanye ngaphezulu ngaphambi kokuba uve isibonelelo esipheleleyo se-ziprasidone. Qhubeka uthathe i-ziprasidone nokuba uziva uphilile. Ungayeki ukuthatha i-ziprasidone ngaphandle kokuthetha nogqirha wakho.

Eli yeza linokumiselwa ezinye izinto; buza ugqirha wakho okanye usokhemesti ngolwazi oluthe kratya.

Ngaphambi kokuba uthathe i-ziprasidone,

  • xelela ugqirha wakho kunye nosokhemisti ukuba ngaba uxabisa i-ziprasidone, nawaphi na amanye amayeza, okanye naziphi na izithako kwiifomsile ze-ziprasidone. Buza usokhemesti wakho uluhlu lwezithako.
  • xelela ugqirha wakho ukuba uthatha i-amiodarone (Cordarone, Pacerone), arsenic trioxide (Trisenox), chlorpromazine, disopyramide (Norpace), dofetilide (Tikosyn), dolasetron (Anzemet), dronedarone (Multaq), droperidol (Inapsine), gatiflo ifumaneka kwi-US), halofantrine (Halfan) (ayisekho e-US), ibutilide (Corvert), levomethadyl (ORLAAM) (ayisekho e-US), mefloquine, mesoridazine (ayisafumaneki e-US), moxifloxacin (Avelox), pentamidine (NebuPent, Pentam), pimozide (Orap), probucol (engasekhoyo e-US), procainamide, quinidine (eNuedexta), sotalol (Betapace, Sorine, Sotylize), sparfloxacin (ayisafumaneki i-US), itacrolimus (Astagraf, Prograf), okanye thioridazine. Ugqirha wakho unokukuxelela ukuba ungathathi i-ziprasidone ukuba uthatha elinye okanye ngaphezulu kula mayeza. Amanye amayeza anokusebenzisana ne-ziprasidone, ke qiniseka ukuxelela ugqirha wakho ngawo onke amayeza owathathayo, nkqu nalawo angaveli kolu luhlu.
  • xelela ugqirha wakho kunye nosokhemesti ukuba loluphi olunye amayeza amiselweyo kunye nalawo angabhalwanga, iivithamini, izongezo zesondlo, kunye nemveliso yamayeza owathathayo okanye oceba ukuyithatha. Qiniseka ukuba ukhankanya nayiphi na kwezi zinto zilandelayo: amayeza oxinzelelo; carbamazepine (Carbatrol, Tegretol, Teril, nabanye); umchamo ('iipilisi zamanzi'); Iidopamine agonists ezinje ngebromocriptine (ICycloset, Parlodel), icabergoline, levodopa (eSinemet), igolide (iPermax) (engasafumaneki e-U.S), kunye ne-ropinirole (i-Requip); ketoconazole (Nizoral); amayeza oxinzelelo lwegazi oluphezulu, ukugula ngengqondo, ukuxhuzula, okanye unxunguphalo; kunye nokuthomalalisa, iipilisi zokulala, okanye iziqandisi. Ugqirha wakho unokufuna ukutshintsha amayeza akho okanye akubeke esweni ngononophelo kwiziphumo ebezingalindelekanga.
  • xelela ugqirha wakho ukuba unokusilela kwentliziyo, isifo seQT eside (imeko yentliziyo enokubangela ukuba nesiyezi, ukuphelelwa ngamandla, okanye ukubetha kwentliziyo ngendlela engaqhelekanga), okanye ukuba ubusandula ukuba nesifo sentliziyo. Ugqirha wakho uya kukuxelela ukuba ungathathi i-ziprasidone.
  • xelela ugqirha wakho ukuba ukhe wazibuza okanye uzikhathaze ngokuzibulala, umhlaza webele, ukubetha kwentliziyo okungaqhelekanga, ukubetha okanye i-ministroke, ukuxhuzula, isifo seswekile, idyslipidemia (amanqanaba aphezulu e-cholesterol), unengxaki yokugcina ibhalansi yakho, okanye isifo sentliziyo okanye sesibindi. Kwakhona, xelela ugqirha wakho ukuba amanqanaba asezantsi e-potassium okanye i-magnesium egazini lakho, ukuba usebenzisa okanye wakha wasebenzisa iziyobisi ezitalatweni okanye wasebenzisa kakhulu amayeza kagqirha, okanye unengxaki yokuginya. Xelela ugqirha wakho ukuba unorhudo okanye ukugabha kakhulu okanye ucinga ukuba unamanzi emzimbeni.
  • xelela ugqirha wakho ukuba ukhulelwe, ngakumbi ukuba ukwinyanga ezimbalwa ezidlulileyo zokukhulelwa kwakho, okanye ukuba ucwangcisa ukukhulelwa okanye ukuncancisa. Ukuba ukhulelwa ngelixa uthatha i-ziprasidone, tsalela ugqirha wakho. I-Ziprasidone inokubangela iingxaki kwiintsana ezisandula ukuzalwa emva kokubeleka ukuba ithathwa ngeenyanga zokugqibela zokukhulelwa. Akufanele uncelise xa uthatha i-ziprasidone.
  • Kuya kufuneka uyazi ukuba i-ziprasidone inokukwenza wozele. Musa ukuqhuba imoto okanye usebenzise oomatshini de ube uyazi indlela elikuchaphazela ngayo eli yeza.
  • Kuya kufuneka uyazi ukuba utywala bunokongeza ukozela okubangelwa leli yeza. Musa ukusela utywala ngelixa uthatha i-ziprasidone.
  • Kuya kufuneka uyazi ukuba unokufumana i-hyperglycemia (inyuka kwiswekile esegazini lakho) ngelixa uthatha eli yeza, nokuba awukabinaso isifo seswekile. Ukuba une-schizophrenia, kunokwenzeka ukuba ube nesifo seswekile kunabantu abangenayo i-schizophrenia, kwaye ukuthatha i-ziprasidone okanye amayeza afanayo kunokuwunyusa lo mngcipheko. Tshela ugqirha wakho kwangoko ukuba unayo nayiphi na le mpawu ilandelayo ngelixa uthatha i-ziprasidone: ukunxanwa okugqithisileyo, ukuchama rhoqo, indlala egqithisileyo, umbono ophuthileyo, okanye ubuthathaka. Kubaluleke kakhulu ukubiza ugqirha wakho nje ukuba ube nazo naziphi na ezi mpawu, kuba iswekile ephezulu yegazi enganyangekiyo inokubangela imeko embi ebizwa ngokuba yi ketoacidosis. I-Ketoacidosis inokuba sengozini yobomi ukuba ayinyangwa kwangoko. Iimpawu zeketoacidosis zibandakanya umlomo owomileyo, isicaphucaphu kunye nokugabha, ukuphefumla kancinci, ukuphefumla okunuka iziqhamo kunye nokuncipha kwengqondo.
  • Kuya kufuneka uyazi ukuba i-ziprasidone inokubangela ukuba ube nesiyezi, ukuba nentloko elula, kunye nokuphelelwa ngamandla xa usukuma ngokukhawuleza kwindawo olele kuyo. Oku kuqheleke ngakumbi xa uqala ukuthatha i-ziprasidone.Ukuthintela le ngxaki, phuma kancinci ebhedini, uphumle iinyawo zakho phantsi imizuzu embalwa ngaphambi kokuba ume.
  • Kuya kufuneka uyazi ukuba i-ziprasidone inokwenza kube nzima ukuba umzimba wakho uphole xa kushushu kakhulu. Tshela ugqirha wakho ukuba ucwangcisa ukwenza umthambo ngamandla okanye uvezwe bubushushu obugqithisileyo.

Thetha nogqirha wakho malunga nokutya igrapefruit kunye nokusela ijusi yegrapefruit ngelixa uthatha eli yeza.


Thatha idosi ephosiweyo ngokukhawuleza nje ukuba uyikhumbule. Nangona kunjalo, ukuba phantse lixesha ledosi elandelayo, tsiba idosi ephosiweyo kwaye uqhubeke neshedyuli yakho yethamo eqhelekileyo. Sukuthatha idosi ephindwe kabini ukwenza eyilahlekileyo.

I-Ziprasidone inokubangela iziphumo ebezingalindelekanga. Tshela ugqirha wakho ukuba ngaba ezinye zeempawu zinzima okanye azihambi:

  • intloko ebuhlungu
  • ukungazinzi
  • ixhala
  • ukunqongophala kwamandla
  • ukuqhina
  • urhudo
  • Ukuphelelwa ngumdla wokutya
  • iintlungu zemisipha
  • isisu esibuhlungu
  • impumlo enemifinya
  • ukukhohlela
  • ukutyeba kwakho
  • ukwandiswa kwamabele okanye ukukhupha
  • ukuya emva kwexesha okanye ukuphoswa lixesha lokuya exesheni
  • ukunciphisa amandla esini
  • isiyezi, ukuziva ungazinzanga, okanye unengxaki yokugcina ibhalansi yakho

Ezinye iziphumo ebezingalindelekanga zinokuba nzulu. Ukuba ufumana naziphi na kwezi mpawu zilandelayo okanye ezo zidweliswe kwicandelo LESILUMKISO ESIBALULEKILEYO okanye icandelo LOKULUMKELA OKUKHETHEKILEYO, tsalela umnxeba kwangoko okanye ufumane unyango olungxamisekileyo:

  • iintshukumo ezingaqhelekanga zobuso bakho okanye zomzimba ongenakuzilawula
  • ngokukhawuleza, ngokungaqhelekanga, okanye ukubetha kwentliziyo
  • irhashalala okanye urticaria
  • ukurhawuzelela
  • i-blisters okanye ukuxobuka kwesikhumba
  • izilonda zomlomo
  • amadlala adumbileyo
  • ifiva
  • Ukugodola
  • ndingcangcazela
  • ukuqina kwemisipha
  • ukuwa
  • ukudideka
  • ukubila
  • ukulahleka kwengqondo
  • ukwakhiwa okubuhlungu kwepenisi okuhlala iiyure

I-Ziprasidone inokubangela ezinye iziphumo ebezingalindelekanga. Biza ugqirha wakho ukuba unengxaki engaqhelekanga ngelixa uthatha eli yeza.


Ukuba uhlangabezana neziphumo ebezingalindelekanga ezimandundu, wena okanye ugqirha wakho ungathumela ingxelo kwiNkqubo yoKutya kunye nezoLawulo (i-FDA) yeMedWatch yeNkqubo yokuNgxelo ngezeMeko eziGwenxa kwi-Intanethi (http://www.fda.gov/Safety/MedWatch) okanye ngomnxeba ( 1-800-332-1088).

Gcina eli yeza kwisikhongozeli lifikile, livalekile, kwaye alifumaneki ebantwaneni. Yigcine kubushushu begumbi kude nokukhanya kunye nobushushu obungaphezulu kunye nobumanzi (hayi kwigumbi lokuhlambela).

Kubalulekile ukugcina onke amayeza ngaphandle kwamehlo kunye nokufikelela kwabantwana njengezikhongozeli ezininzi (ezinje ngeeveki zeepilisi zeveki kunye nezo zamehlo, iikhrim, iipatches, kunye ne-inhalers) azinyangeki kwaye abantwana abancinci banokuzivula ngokulula. Ukukhusela abantwana abancinci kwiityhefu, soloko ukhiya iminqwazi yokhuseleko kwaye ubeke amayeza kwindawo ekhuselekileyo-leyo iphakame kwaye iphakame kwaye ingabonakali kubo kwaye ifikelele kuyo. http://www.upandaway.org

Amayeza angafunekiyo kufuneka achithwe ngeendlela ezizodwa zokuqinisekisa ukuba izilwanyana zasekhaya, abantwana kunye nabanye abantu abanakuzisebenzisa. Nangona kunjalo, akufuneki uligungxule eli yeza kwindlu yangasese. Endaweni yoko, eyona ndlela yokulahla amayeza akho yinkqubo yokubuyisa amayeza. Thetha kumayeza wakho okanye unxibelelane nesebe lakho lenkunkuma / lokurisayikilisha ukuze ufunde malunga neenkqubo zokubuyisa kwindawo ohlala kuyo. Jonga i-FDA's Safe Disposal of Medicines website (http://goo.gl/c4Rm4p) ngolwazi oluthe kratya ukuba awunakho ukufikelela kwinkqubo yokubuyisa.

Kwimeko yokugqithisa, fowunela umnxeba wolawulo lwetyhefu kwi-1-800-222-1222. Ulwazi lukwafumaneka kwi-Intanethi kwi-https: //www.poisonhelp.org/help. Ukuba ixhoba liye lawa, laxhuzula, linengxaki yokuphefumla, okanye alikwazi ukuvuswa, ngoko nangoko lifowunele iinkonzo zongxamiseko ngo-911.

Iimpawu libanda kungaquka oku kulandelayo:

  • ukozela
  • intetho engacacanga
  • iintshukumo ngequbuliso ongenakuzilawula
  • ukushukuma okungalawulekiyo kwilungu lomzimba
  • ixhala

Gcina lonke ixesha lokudibana nogqirha wakho kunye nelabhoratri. Ugqirha wakho angayalela iimvavanyo ezithile zebhu ukujonga impendulo yomzimba wakho kwi-ziprasidone.

Musa ukuvumela nabani na ukuba athathe amayeza akho. Buza usokhemesti wakho nayiphi na imibuzo onayo malunga nokuzalisa amayeza akho.

Kubalulekile ukuba ugcine uluhlu olubhaliweyo lwawo onke amayeza owasebenzisayo amayeza owasebenzisayo, kunye nezinye iimveliso ezinjengeevithamini, iiminerali, okanye ezinye izongezo zokutya. Kuya kufuneka uze nolu luhlu qho xa undwendwela ugqirha okanye ungeniswe esibhedlele. Kukwabalulekile ulwazi ukuba uphathe nawe xa kukho imeko kaxakeka.

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